SCHEMBL7410551

SCHEMBL7410551

CC(C)(C)OC(=O)N(NC(=O)c1cccc(NC(=N)N)c1)[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.41
ITGA2B P08514 2/20 0.41
ITGB1 P05556 1/20 0.41
ITGAV P06756 1/20 0.41
ITGB5 P18084 1/20 0.41
BACE1 P56817 2/20 0.40
SLC7A5 Q01650 1/20 0.39
F2 P00734 5/20 0.38
TMPRSS6 Q8IU80 2/20 0.38
CASR P41180 1/20 0.37
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
LMNA P02545 1/20 0.37
KCNK3 O14649 1/20 0.36
KCNK9 Q9NPC2 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
MAPT P10636 1/20 0.36
NTSR1 P30989 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410381 1.00 ITGB3 (0.41) ITGB3ITGA2BITGB1ITGAVITGB5
Phenylalanine SCHEMBL7414620 0.96 SLC7A5 (0.47) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7408424 0.91 ALDH1A1 (0.41) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7375593 0.91 ALDH1A1 (0.42) ITGB3ITGA2BF2CASRLMNA
SCHEMBL7466483 0.88 NPC1 (0.45) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7409600 0.88 MAPT (0.42) LMNANR1H4MAPTNPSR1MEN1
SCHEMBL7382269 0.86 NR1H4 (0.41) ITGB3ITGA2BITGAVF2LMNA
SCHEMBL7376793 0.86 RAB9A (0.38) ITGB3ITGA2BF2LMNAMAPT
SCHEMBL7410561 0.86 ITGB3 (0.40) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7410389 0.86 ITGB3 (0.40) ITGB3ITGA2BITGB1ITGAVITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed