SCHEMBL7376017

SCHEMBL7376017

Cc1cc(-c2ccccc2)c(Cl)cc1[C]=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
CYP2A6 P11509 2/20 0.39
PRKAG1 P54619 5/20 0.38
PRKAA2 P54646 5/20 0.38
PRKAB1 Q9Y478 5/20 0.38
PRKAB2 O43741 4/20 0.38
PRKAA1 Q13131 4/20 0.38
PRKAG3 Q9UGI9 4/20 0.38
PRKAG2 Q9UGJ0 4/20 0.38
CSNK2A1 P68400 2/20 0.38
ESR2 Q92731 1/20 0.37
KDM4E B2RXH2 2/20 0.36
HPGD P15428 2/20 0.36
GALR3 O60755 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
HSD11B1 P28845 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7370563 0.83 SRD5A2 (0.49) PRKAG1PRKAA2PRKAB1PRKAB2PRKAA1
SCHEMBL7371062 0.81 BACE1 (0.52) CYP2A6ESR2KDM4EHPGDGALR3
SCHEMBL7374419 0.79 LMNA (0.40) NPSR1CYP1A2CYP2C9CYP2C19CYP2A6
SCHEMBL27142057 0.79 CYP2A6 (0.50) NPSR1CYP1A2CYP2C9CYP2C19CYP2A6
SCHEMBL7375894 0.77 PGR (0.46) CYP1A2CYP2C9CYP2C19CYP2A6KDM4E
SCHEMBL7368661 0.76 AR (0.41) ESR2KDM4EHPGDGALR3ALDH1A1
SCHEMBL7368488 0.73 ALDH1A1 (0.35) NPSR1CYP1A2CYP2C9CYP2C19CYP2A6
SCHEMBL26606940 0.73 BACE1 (0.50) NPSR1CYP1A2CYP2C9CYP2C19CYP2A6
SCHEMBL27517035 0.72 GABRA1 (0.46) CYP1A2CYP2C9CYP2C19KDM4EHPGD
SCHEMBL5885406 0.71 CYP2A6 (0.50) CYP2A6PRKAG1PRKAA2PRKAB1PRKAB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994021650-A1 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-09-29 WO disclosed