SCHEMBL7376402

SCHEMBL7376402

COc1cc(C(=O)N(C)C)cc(OC)c1OC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB4A P04350 3/20 0.51
TUBB P07437 3/20 0.51
TUBA3C P0DPH7 3/20 0.51
TUBA1B P68363 3/20 0.51
TUBA4A P68366 3/20 0.51
TUBB4B P68371 3/20 0.51
TUBB3 Q13509 3/20 0.51
TUBB2A Q13885 3/20 0.51
TUBB8 Q3ZCM7 3/20 0.51
TUBA3E Q6PEY2 3/20 0.51
TUBA1A Q71U36 3/20 0.51
TUBA1C Q9BQE3 3/20 0.51
TUBB6 Q9BUF5 3/20 0.51
TUBB2B Q9BVA1 3/20 0.51
TUBB1 Q9H4B7 3/20 0.51
ALDH1A1 P00352 4/20 0.50
MAPT P10636 3/20 0.50
LMNA P02545 2/20 0.50
MAPK1 P28482 1/20 0.50
GFER P55789 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7384060 0.87 SCN1A (0.45) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL1436447 0.86 TUBB4A (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL709048 0.85 ABCG2 (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL1004147 0.84 RXFP1 (0.53) ALDH1A1LMNATPMTKMT2AMEN1
SCHEMBL2486085 0.84 PKM (0.62) ALDH1A1MAPTLMNAMAPK1KMT2A
SCHEMBL11229430 0.82 ALDH1A1 (0.46) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL1003355 0.80 BRD4 (0.44) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL9545203 0.79 HSP90AA1 (0.61) ALDH1A1MAPK1SCN1ASCN2ASCN3A
SCHEMBL7276036 0.79 KMT2A (0.49) ALDH1A1MAPTLMNAMAPK1GFER
SCHEMBL4625442 0.79 TUBB1 (0.58) TUBB4ATUBBTUBA3CTUBA1BTUBA4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6486155-B1 Method of inhibiting neoplastic cells with isoquinoline derivatives CELL PATHWAYS INC 2002-11-26 US disclosed
WO-1998038168-A1 ISOQUINOLINONE DERIVATIVES, PROCESS FOR PREPARING THE SAME, AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS TANABE SEIYAKU CO., LTD. (JP) 1998-09-03 WO disclosed