SCHEMBL7379264

SCHEMBL7379264

O=[C]c1cccc(NC(=O)c2ccccc2)c1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 8/20 0.71
KCNK9 Q9NPC2 6/20 0.71
SIRT1 Q96EB6 2/20 0.68
RAB9A P51151 4/20 0.61
NPC1 O15118 3/20 0.61
HPGD P15428 1/20 0.61
KMT2A Q03164 5/20 0.59
MEN1 O00255 4/20 0.59
TP53 P04637 1/20 0.59
POLB P06746 2/20 0.58
NLRP3 Q96P20 1/20 0.56
HPSE Q9Y251 1/20 0.56
ALDH1A1 P00352 1/20 0.55
MAPT P10636 1/20 0.55
LPAR3 Q9UBY5 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11596555 0.86 KCNK3 (0.59) KCNK3KCNK9SIRT1RAB9ANPC1
SCHEMBL2173418 0.85 HTT (0.71) KCNK3KCNK9SIRT1RAB9ANPC1
SCHEMBL5612900 0.85 KCNK3 (0.69) KCNK3KCNK9SIRT1RAB9ANPC1
SCHEMBL2298254 0.84 KCNK3 (1.00) KCNK3KCNK9SIRT1RAB9ANPC1
SCHEMBL1680201 0.81 KCNK3 (0.50) KCNK3KCNK9SIRT1RAB9ANPC1
SCHEMBL9799718 0.81 PTGS1 (0.60) KCNK3KCNK9SIRT1KMT2AMEN1
SCHEMBL363342 0.81 PTPN1 (0.67) KCNK3KCNK9SIRT1RAB9ANPC1
SCHEMBL19491390 0.81 SIRT1 (1.00) KCNK3KCNK9SIRT1RAB9ANPC1
SCHEMBL363881 0.81 PTPN1 (0.67) KCNK3KCNK9SIRT1RAB9ANPC1
SCHEMBL14715827 0.80 KCNK3 (0.92) KCNK3KCNK9SIRT1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087946-A1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2001-04-04 EP disclosed
WO-1999065880-A1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GMBH (DE) 1999-12-23 WO disclosed