SCHEMBL7388341

SCHEMBL7388341

CN(C(=O)C[C@H](NC(=O)OCc1ccccc1)C(=O)N(CCC(=O)O)C1CC1)[C@H]1CCCN(C(=N)N)C1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.41
CASP1 P29466 1/20 0.41
ITGB3 P05106 2/20 0.40
ITGA2B P08514 2/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
CTSL P07711 3/20 0.40
CTSS P25774 3/20 0.40
CTSB P07858 1/20 0.40
OPRK1 P41145 1/20 0.40
ACE P12821 1/20 0.40
IL2RA P01589 1/20 0.39
ALB P02768 1/20 0.39
IL2 P60568 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
F10 P00742 1/20 0.39
PRSS1 P07477 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7397245 0.93 CASP1 (0.41) CTSKCASP1ADORA3ADORA2AADORA2B
Hydrochloric Acid SCHEMBL9002984 0.92 CASP1 (0.41) CTSKCASP1ADORA3ADORA2AADORA2B
SCHEMBL7392968 0.90 ITGB3 (0.39) CTSKCASP1ITGB3ITGA2BADORA3
SCHEMBL7395541 0.88 CTSK (0.40) CTSKCASP1ADORA3ADORA2AADORA2B
SCHEMBL7393462 0.87 L3MBTL1 (0.38) CTSKCASP1ITGB3ITGA2BADORA3
Hydrochloric Acid SCHEMBL9003066 0.86 L3MBTL1 (0.38) CTSKCASP1ITGB3ITGA2BADORA3
SCHEMBL9003040 0.84 F2 (0.47) ITGB3ITGA2BIL2RAALBIL2
SCHEMBL7391071 0.84 TPSAB1 (0.40) ACEL3MBTL1PRSS1
Hydrochloric Acid SCHEMBL9002664 0.83 TPSAB1 (0.40) ACEL3MBTL1PRSS1
SCHEMBL7395266 0.82 CASP1 (0.40) CTSKCASP1ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5559232-A ANTICOAGULANTS HOFFMANN-LA ROCHE INC. (US) 1996-09-24 US disclosed
EP-0641779-A1 Novel 1-amidinopiperdines and 4-amidinomorpholines as aggregation inhibitions F. HOFFMANN-LA ROCHE AG (CH) 1995-03-08 EP disclosed