SCHEMBL7393237

SCHEMBL7393237

CN(CC(Cc1ccccc1)C(=O)O)C(=O)OCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.53
ABCB1 P08183 2/20 0.49
CPA1 P15085 6/20 0.47
CPA3 P15088 3/20 0.47
FOLH1 Q04609 1/20 0.47
CPB1 P15086 1/20 0.47
CPB2 Q96IY4 1/20 0.47
SLC15A1 P46059 1/20 0.47
ALDH1A1 P00352 2/20 0.46
ACE2 Q9BYF1 1/20 0.45
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
SLC1A3 P43003 1/20 0.44
SLC1A2 P43004 1/20 0.44
SLC1A1 P43005 1/20 0.44
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14405551 0.83 SLC15A1 (0.42) ABCB1SLC15A1ALDH1A1ACE2ITGB3
SCHEMBL13687217 0.82 ALDH1A1 (0.51) ABCB1ALDH1A1MAPTHPGD
SCHEMBL23699429 0.82 CYP1A2 (0.51) CYP1A2CPA1CPA3FOLH1CPB1
SCHEMBL2968658 0.79 ITGB3 (0.59) ABCB1FOLH1ALDH1A1ITGB3ITGA2B
SCHEMBL31739224 0.79 ITGB3 (0.59) ABCB1FOLH1ALDH1A1ITGB3ITGA2B
SCHEMBL2494968 0.79 ITGB3 (0.59) ABCB1FOLH1ALDH1A1ITGB3ITGA2B
SCHEMBL8067076 0.79 ITGB3 (0.59) ABCB1FOLH1ALDH1A1ITGB3ITGA2B
SCHEMBL358090 0.79 ALDH1A1 (0.49) ABCB1ALDH1A1MAPTHPGD
SCHEMBL19541343 0.79 ALDH1A1 (0.49) CYP1A2ABCB1SLC15A1ALDH1A1SLC1A3
SCHEMBL26654515 0.78 ITGB3 (0.58) ABCB1FOLH1ALDH1A1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0670310-B1 Bisulfite adducts of arginine aldehydes useful as thrombin inhibitors and as anticoagulants LILLY CO ELI (US) 1998-09-02 EP disclosed
US-5488037-A ARGININE ALDEHYDE DERIVATIVES ELI LILLY AND COMPANY (US) 1996-01-30 US disclosed
EP-0671390-A2 Antithrombotic agents ELI LILLY AND COMPANY (US) 1995-09-13 EP disclosed
EP-0670310-A1 Bisulfite adducts of arginine aldehydes useful as thrombin inhibitors and as anticoagulants ELI LILLY AND COMPANY (US) 1995-09-06 EP disclosed
US-5436229-A Di- and tripeptides as anticoagulants ELI LILLY AND COMPANY (US) 1995-07-25 US disclosed