SCHEMBL23699429

SCHEMBL23699429

CN(CC(Cc1ccccc1)C(=O)O)C(=O)OC(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.51
CPA1 P15085 7/20 0.46
CPA3 P15088 3/20 0.46
FOLH1 Q04609 2/20 0.46
CPB1 P15086 1/20 0.46
CPB2 Q96IY4 1/20 0.46
SLC1A3 P43003 1/20 0.43
SLC1A2 P43004 1/20 0.43
SLC1A1 P43005 1/20 0.43
HTR2C P28335 1/20 0.42
SLC6A4 P31645 1/20 0.42
ATM Q13315 1/20 0.42
ITGA4 P13612 1/20 0.42
ITGB7 P26010 1/20 0.42
ACE P12821 1/20 0.42
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16798442 0.88 CTSS (0.44) CYP1A2CPA1ACE
SCHEMBL16798328 0.88 KMT2A (0.43) CYP1A2
SCHEMBL23719091 0.88 CTSK (0.44) HTR2CSLC6A4ACE
SCHEMBL23699255 0.88 CTSK (0.44) HTR2CSLC6A4ACE
SCHEMBL18116069 0.87 CYP1A2 (0.53) CYP1A2CPA1CPA3FOLH1CPB1
SCHEMBL16798383 0.87 LDHA (0.51)
SCHEMBL23699444 0.86 FOLH1 (0.50) CYP1A2CPA1CPA3FOLH1CPB1
SCHEMBL23699358 0.86 CTSS (0.47) FOLH1SLC1A1HTR2CSLC6A4ATM
SCHEMBL23699341 0.85 PPARA (0.45) CYP1A2FOLH1
SCHEMBL23699431 0.85 MAOB (0.42) FOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3858439-A1 AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN ESTEVE PHARMACEUTICALS, S.A. (ES) 2021-08-04 EP disclosed
EP-3858439-A1 AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN ESTEVE PHARMACEUTICALS, S.A. (ES) 2021-08-04 EP disclosed