SCHEMBL7397186

SCHEMBL7397186

COc1ccc(N2CCN(C(=O)CC3CCCc4ccccc43)CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.54
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
UGCG Q16739 1/20 0.52
MAPT P10636 4/20 0.52
ALDH1A1 P00352 2/20 0.52
LMNA P02545 2/20 0.52
GFER P55789 2/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
PKM P14618 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7403392 0.94 MAPK1 (0.56) MAPK1MEN1KMT2AMAPTALDH1A1
SCHEMBL7404596 0.83 DRD2 (0.59) MAPK1MEN1KMT2AMAPTALDH1A1
SCHEMBL7397389 0.80 DRD4 (0.66)
SCHEMBL9014716 0.79 HTR1A (0.47) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL7402337 0.79 DRD2 (0.48) MEN1KMT2AUGCGMAPTALDH1A1
Hydrochloric Acid SCHEMBL7399648 0.79 DRD4 (0.64)
SCHEMBL7402692 0.78 MAPK1 (0.55) MAPK1MEN1KMT2AMAPTALDH1A1
Hydrochloric Acid SCHEMBL7398492 0.78 DRD2 (0.48) MAPK1MEN1KMT2AUGCGMAPT
SCHEMBL8347285 0.76 MTNR1B (0.61) MAPK1MAPTALDH1A1HPGDHSD17B10
SCHEMBL27529224 0.76 MTNR1B (0.61) MAPK1MAPTALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6133446-A Heterocyclic compounds for the treatment of CNS and cardiovascular disorders PHARMACIA & UPJOHN COMPANY (US) 2000-10-17 US disclosed
WO-1995018118-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF CNS AND CARDIOVASCULAR DISORDERS THE UPJOHN COMPANY (US) 1995-07-06 WO disclosed