SCHEMBL7397635

SCHEMBL7397635

COC(=O)c1ccc(C(=O)Oc2cccc3[nH]nnc23)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 1/20 0.44
LMNA P02545 5/20 0.42
POLB P06746 1/20 0.42
RAB9A P51151 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 3/20 0.42
KMT2A Q03164 3/20 0.42
NPC1 O15118 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 1/20 0.42
TP53 P04637 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.42
MAPT P10636 4/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
KDM4E B2RXH2 2/20 0.41
AR P10275 1/20 0.41
PKM P14618 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6155017 0.87 LMNA (0.54) SLC6A3LMNAPOLBKMT2ASMN1; SMN2
SCHEMBL8827881 0.84 LMNA (0.39) LMNAPOLBALDH1A1KMT2ASMN1; SMN2
SCHEMBL7707716 0.80 SLC22A6 (0.44) LMNAPOLBRAB9AALDH1A1HPGD
SCHEMBL8844752 0.79 MAPT (0.33) LMNAPOLBMAPTKDM4EMETAP2
SCHEMBL44289 0.79 MAPT (0.33) LMNAPOLBHPGDMAPTKDM4E
SCHEMBL7403840 0.79 GAA (0.47) LMNAPOLBALDH1A1KMT2ASMN1; SMN2
SCHEMBL44290 0.78 LMNA (0.35) LMNAPOLBALDH1A1KMT2AMEN1
SCHEMBL14690221 0.77 MAPT (0.32) LMNAPOLBMAPTKDM4EMETAP2
SCHEMBL717583 0.77 PKN1 (0.50) LMNAPOLBALDH1A1KMT2AMAPT
SCHEMBL2534586 0.77 MEN1 (0.38) LMNAPOLBKMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255748-A1 BETA-ALANINE DERIVATIVES AND THEIR USE AS RECEPTOR ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-11-13 EP disclosed
WO-2001060813-A1 BETA-ALANINE DERIVATIVES AND THEIR USE AS RECEPTOR ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-08-23 WO disclosed