SCHEMBL7399114

SCHEMBL7399114

COC(=O)c1sccc1N(C(=O)OC(C)(C)C)C1CCNCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
ALDH1A1 P00352 5/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
CASP3 P42574 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NPC1 O15118 1/20 0.37
HTT P42858 1/20 0.36
RXFP1 Q9HBX9 2/20 0.35
TSHR P16473 2/20 0.35
KDM4E B2RXH2 2/20 0.35
CYP1A2 P05177 1/20 0.34
POLB P06746 1/20 0.34
PRNP P04156 1/20 0.34
MAPK10 P53779 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399731 0.88 LMNA (0.35) KMT2AMEN1ALDH1A1GAAL3MBTL1
SCHEMBL2873412 0.79 ALDH1A1 (0.41) KMT2AMEN1ALDH1A1SMN1; SMN2GAA
SCHEMBL2873409 0.79 ALDH1A1 (0.41) KMT2AMEN1ALDH1A1SMN1; SMN2GAA
SCHEMBL4729037 0.76 NPC1 (0.47) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL22261640 0.75 NPC1 (0.46) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8437522 0.75 SLC6A2 (0.38) KMT2AMEN1CYP2D6SLC6A2SLC6A4
SCHEMBL4439262 0.74 EPHX2 (0.39) KMT2AMEN1ALDH1A1SMN1; SMN2SLC6A2
SCHEMBL5214565 0.74 SLC6A2 (0.37) KMT2AMEN1CYP2D6SLC6A2SLC6A4
SCHEMBL7399910 0.74 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3
SCHEMBL12469312 0.73 SLC6A2 (0.46) KMT2AMEN1ALDH1A1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714299-A4 1996-07-10 EP disclosed
EP-0714299-A1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO. INC. (US) 1996-06-05 EP disclosed
WO-1995002405-A1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1995-01-26 WO disclosed