SCHEMBL7399686

SCHEMBL7399686

CC(CCC(=O)NCC#N)Cc1cccc(-c2cccc(C#N)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSS P25774 12/20 0.47
CTSL P07711 10/20 0.47
CTSB P07858 9/20 0.47
CTSK P43235 3/20 0.47
MME P08473 1/20 0.44
CTSV O60911 5/20 0.43
MMP12 P39900 1/20 0.42
MMP13 P45452 1/20 0.42
FOLH1 Q04609 1/20 0.41
MCHR1 Q99705 2/20 0.40
GPR139 Q6DWJ6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7401952 0.92 CTSS (0.51) CTSSCTSLCTSBCTSKMME
SCHEMBL7400496 0.85 CTSS (0.60) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7395140 0.84 CTSS (0.44) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7405777 0.83 CTSL (0.45) CTSSCTSLCTSBCTSKMME
SCHEMBL7401735 0.82 CTSS (0.48) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7397511 0.81 CTSL (0.51) CTSSCTSLCTSBCTSK
SCHEMBL7441160 0.81 CTSS (0.43) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7394745 0.80 CTSL (0.59) CTSSCTSLCTSBCTSK
SCHEMBL7392809 0.80 NTSR1 (0.45) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7447689 0.80 CTSS (0.43) CTSSCTSLCTSBCTSKCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001049288-A9 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2001-10-25 WO disclosed