SCHEMBL7405458

SCHEMBL7405458

COCCOCCOCCOc1ccc2c(O)c(C(c3cccc(N4C=CN(C)C4)c3)C3CC3)c(=O)oc2c1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.36
ACHE P22303 3/20 0.35
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
PRKDC P78527 1/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400115 0.84 ACHE (0.40) ACHEPRKDC
SCHEMBL7405459 0.78 HDAC1 (0.34) SIGMAR1ACHEPRKDC
SCHEMBL7400677 0.77 ROCK2 (0.35) ACHE
SCHEMBL7400973 0.77 MAOB (0.40) ACHE
SCHEMBL7403592 0.76 NQO1 (0.36) ACHE
SCHEMBL7405503 0.74 FABP1 (0.44) TP53POLB
SCHEMBL7359563 0.73 CYP2C9 (0.58) ACHE
SCHEMBL7354182 0.67 NQO1 (0.42) POLB
SCHEMBL8868342 0.66 NQO1 (0.49) TP53POLB
SCHEMBL7403259 0.65 MEN1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030670-A2 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-16 WO disclosed