SCHEMBL7405459

SCHEMBL7405459

COCCOCCOCCOc1ccc2c(O)c(C(c3cccc([N+]4(C)C=CN=C4)c3)C3CC3)c(=O)oc2c1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.34
ACHE P22303 5/20 0.33
MAP1LC3B Q9GZQ8 1/20 0.33
MAP1LC3A Q9H492 1/20 0.33
APP P05067 1/20 0.33
BCHE P06276 1/20 0.32
PRKDC P78527 1/20 0.32
NQO1 P15559 3/20 0.32
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400115 0.83 ACHE (0.40) HDAC1ACHEMAP1LC3BMAP1LC3APRKDC
SCHEMBL7405458 0.78 SIGMAR1 (0.36) ACHEPRKDCSIGMAR1
SCHEMBL7400973 0.78 MAOB (0.40) ACHEMAP1LC3BMAP1LC3ANQO1
SCHEMBL7403592 0.76 NQO1 (0.36) ACHEMAP1LC3BMAP1LC3ANQO1
SCHEMBL7400677 0.75 ROCK2 (0.35) ACHE
SCHEMBL7405503 0.74 FABP1 (0.44) MAP1LC3BMAP1LC3A
SCHEMBL7359563 0.73 CYP2C9 (0.58) ACHENQO1
SCHEMBL7354182 0.66 NQO1 (0.42) NQO1
SCHEMBL8868342 0.66 NQO1 (0.49) NQO1
SCHEMBL7403259 0.63 MEN1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030670-A2 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-16 WO disclosed