SCHEMBL7400340

SCHEMBL7400340

COc1cc(-c2nc3cc(C)ccc3[nH]2)ccc1OC(=O)C(C)(C)C

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.59
EPHX2 P34913 1/20 0.59
AMY1A P0DUB6 4/20 0.53
CHEK2 O96017 4/20 0.48
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
PARP1 P09874 2/20 0.45
GUSB P08236 2/20 0.43
PARP2 Q9UGN5 1/20 0.43
PDE4A P27815 3/20 0.42
PDE4B Q07343 3/20 0.42
PDE4C Q08493 3/20 0.42
PDE4D Q08499 3/20 0.42
THRB P10828 1/20 0.41
HPSE Q9Y251 1/20 0.41
SMPD3 Q9NY59 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7388111 0.88 AMY1A (0.66) ALOX5EPHX2AMY1ACHEK2KDM4E
SCHEMBL7386529 0.88 GUSB (0.57) ALOX5EPHX2AMY1ACHEK2KDM4E
SCHEMBL15455607 0.85 ALOX5 (0.80) ALOX5EPHX2AMY1ACHEK2KDM4E
SCHEMBL7391080 0.83 CHEK2 (0.48) CHEK2KDM4EALDH1A1HPSE
SCHEMBL7394125 0.82 AMY1A (0.54) ALOX5EPHX2AMY1AKDM4EALDH1A1
SCHEMBL7389940 0.82 ALDH1A1 (0.71) ALOX5EPHX2AMY1ACHEK2KDM4E
SCHEMBL7396876 0.79 ALOX5 (0.62) ALOX5EPHX2AMY1ACHEK2KDM4E
SCHEMBL7387113 0.78 AMY1A (0.42) AMY1ACHEK2KDM4EALDH1A1HPGD
SCHEMBL7395145 0.77 GUSB (0.47) ALOX5EPHX2AMY1AKDM4EALDH1A1
SCHEMBL22251584 0.77 ACHE (0.57) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1132381-A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them CERMOL S.A. (CH) 2001-09-12 EP claimed
WO-2001066526-A1 ESTER DERIVATIVES OF DIMETHYLPROPIONIC ACID AND PHARMACETUICAL COMPOSITIONS CONTAINING THEM CERMOL S.A. (CH) 2001-09-13 WO disclosed
EP-1132381-A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them CERMOL S.A. (CH) 2001-09-12 EP disclosed