SCHEMBL7388111

SCHEMBL7388111

COc1cc(-c2nc3cc(Cl)ccc3[nH]2)ccc1OC(=O)C(C)(C)C

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 9/20 0.66
ALOX5 P09917 1/20 0.46
EPHX2 P34913 1/20 0.46
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 1/20 0.45
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
PARP1 P09874 2/20 0.44
CHEK2 O96017 2/20 0.44
BRD4 O60885 1/20 0.42
GUSB P08236 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
RHEB Q15382 1/20 0.42
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400340 0.88 ALOX5 (0.59) AMY1AALOX5EPHX2KDM4EALDH1A1
SCHEMBL7386529 0.85 GUSB (0.57) AMY1AALOX5EPHX2KDM4EALDH1A1
SCHEMBL7386703 0.83 CHEK2 (0.48) AMY1AKDM4EALDH1A1HPGDMEN1
SCHEMBL7394125 0.81 AMY1A (0.54) AMY1AALOX5EPHX2KDM4EALDH1A1
SCHEMBL7389940 0.81 ALDH1A1 (0.71) AMY1AALOX5EPHX2KDM4EALDH1A1
SCHEMBL7388752 0.81 KDM4E (0.46) AMY1AKDM4EALDH1A1HPGDMEN1
SCHEMBL7395692 0.79 AMY1A (0.62) AMY1AALOX5EPHX2KDM4EALDH1A1
SCHEMBL7392370 0.79 AMY1A (0.46) AMY1AKDM4EALDH1A1
SCHEMBL7387113 0.77 AMY1A (0.42) AMY1AKDM4EALDH1A1HPGDMEN1
SCHEMBL7397419 0.77 KDM4E (0.52) AMY1AKDM4EALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1132381-A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them CERMOL S.A. (CH) 2001-09-12 EP claimed
WO-2001066526-A1 ESTER DERIVATIVES OF DIMETHYLPROPIONIC ACID AND PHARMACETUICAL COMPOSITIONS CONTAINING THEM CERMOL S.A. (CH) 2001-09-13 WO disclosed
EP-1132381-A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them CERMOL S.A. (CH) 2001-09-12 EP disclosed