SCHEMBL7401699

SCHEMBL7401699

CC(C)[C@H](NS(=O)(=O)CCc1ccncc1)C(=O)N[C@@H](Cc1ccccc1)[C@H](O)[C@@H](O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NS(=O)(=O)CCc1ccncc1)C(C)C

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.51
BACE1 P56817 14/20 0.49
ADAM17 P78536 1/20 0.47
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 1/20 0.43
CTSD P07339 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7332493 1.00 CA2 (0.51) CA2BACE1ADAM17ALDH1A1CYP3A4
SCHEMBL7341693 0.89 CA2 (0.55) CA2BACE1ADAM17
SCHEMBL7332837 0.86 CA2 (0.64) CA2BACE1ALDH1A1CTSD
SCHEMBL7333019 0.86 CA2 (0.64) CA2BACE1ALDH1A1CTSD
SCHEMBL7339716 0.86 CA2 (0.64) CA2BACE1ALDH1A1CTSD
SCHEMBL7358203 0.79 CTSD (0.39) CA2ADAM17CTSD
SCHEMBL7335195 0.79 MMP13 (0.52) ADAM17ALDH1A1
SCHEMBL7335191 0.79 MMP13 (0.52) ADAM17ALDH1A1
SCHEMBL7336565 0.78 ADAM17 (0.46) CA2ADAM17ALDH1A1CYP3A4
SCHEMBL6448985 0.77 CTSD (0.68) CA2BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed