SCHEMBL7401820

SCHEMBL7401820

COC(=O)COc1ccc(C(=O)C(C)Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
PTGS2 P35354 2/20 0.49
MAPT P10636 5/20 0.48
POLB P06746 2/20 0.47
L3MBTL1 Q9Y468 3/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
GAA P10253 2/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3279211 0.87 PTGS2 (0.51) ALDH1A1CYP2C9CYP2C19PTGS2MAPT
SCHEMBL11660766 0.85 ALDH1A1 (0.50) ALDH1A1CYP2C9CYP2C19PTGS2MAPT
SCHEMBL1706669 0.84 ALDH1A1 (0.55) ALDH1A1MAPTKMT2AMEN1SMN1; SMN2
SCHEMBL13846320 0.84 L3MBTL1 (0.43) CYP2C19MAPTL3MBTL1KMT2AGAA
SCHEMBL2116437 0.81 PTGS2 (0.66) ALDH1A1CYP2C9CYP2C19PTGS2MAPT
SCHEMBL23542808 0.81 SMN1; SMN2 (0.57) ALDH1A1GAANPC1RAB9ASMN1; SMN2
SCHEMBL5743825 0.80 PARP10 (0.58) ALDH1A1L3MBTL1KMT2AMEN1GAA
SCHEMBL10299626 0.80 PTGS2 (0.57) ALDH1A1CYP2C9CYP2C19PTGS2MAPT
SCHEMBL4262664 0.78 MAPT (0.70) PTGS2MAPTPOLBL3MBTL1KMT2A
SCHEMBL6960461 0.78 L3MBTL1 (0.61) ALDH1A1CYP2C9CYP2C19PTGS2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5563141-A INHIBIT CELL ADHESION FOR EXAMPLE, PLATELET AGGRE GATION ZENECA LIMITED (GB) 1996-10-08 US disclosed
EP-0690847-A1 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1996-01-10 EP disclosed
WO-1994022835-A2 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1994-10-13 WO disclosed