SCHEMBL7404387

SCHEMBL7404387

CCCCNC(=O)C(Cc1ccccc1)NC(=O)C(CC(C)C)C(=O)NC(C=O)CC(=O)O

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 3/20 0.55
CTSB P07858 1/20 0.52
CASP1 P29466 1/20 0.51
CHRNB2 P17787 1/20 0.48
CHRNB4 P30926 1/20 0.48
CHRNA3 P32297 1/20 0.48
CHRNA4 P43681 1/20 0.48
PTPN1 P18031 1/20 0.48
MMP2 P08253 8/20 0.47
MMP1 P03956 3/20 0.47
MMP3 P08254 3/20 0.47
MMP9 P14780 1/20 0.47
PSMB5 P28074 2/20 0.47
CTSK P43235 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7412065 0.84 CASP1 (0.48) MMP8CTSBCASP1MMP2MMP1
SCHEMBL7404683 0.83 CASP1 (0.59) MMP8CTSBCASP1MMP3MMP9
SCHEMBL7401512 0.83 PLA2G10 (0.43) MMP8CASP1MMP2MMP1MMP3
SCHEMBL7410635 0.81 MMP8 (0.59) MMP8CTSBCASP1MMP3MMP9
SCHEMBL7407874 0.78 MMP8 (0.67) MMP8CTSBCASP1MMP2MMP1
SCHEMBL985563 0.73 CHRNB2 (0.77) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL23086284 0.73 PTPN1 (0.68) CHRNB2CHRNB4CHRNA3CHRNA4PTPN1
SCHEMBL23091304 0.72 PSMB5 (0.64) CTSBPSMB5CTSK
SCHEMBL7411011 0.72 MMP3 (0.53) MMP8CTSBCASP1MMP2MMP1
SCHEMBL7406669 0.72 MMP3 (0.51) MMP8CTSBCASP1MMP2MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed