SCHEMBL740445

SCHEMBL740445

O=C(O)[C@@]1(Cc2ccccc2)CC[C@H]2O[C@H]2C1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
HSD11B1 P28845 1/20 0.35
LMNA P02545 1/20 0.35
MAOA P21397 4/20 0.35
MAOB P27338 4/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
KDM1A O60341 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
GRIN2B Q13224 1/20 0.33
DPP4 P27487 1/20 0.33
GRM6 O15303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1859933 1.00 KDM4E (0.36) KDM4EHSD11B1LMNAMAOAMAOB
SCHEMBL740446 1.00 KDM4E (0.36) KDM4EHSD11B1LMNAMAOAMAOB
SCHEMBL175503 0.77 MAPK1 (0.35) KDM4ELMNASMN1; SMN2
SCHEMBL16005 0.77 MAPK1 (0.35) KDM4ELMNASMN1; SMN2
SCHEMBL923461 0.75 MAOA (0.48) KDM4EHSD11B1LMNAMAOAMAOB
SCHEMBL741407 0.74 MAPK1 (0.37) KDM4ELMNASMN1; SMN2
SCHEMBL741406 0.74 MAPK1 (0.37) KDM4ELMNASMN1; SMN2
SCHEMBL1860545 0.74 MAPK1 (0.37) KDM4ELMNASMN1; SMN2
SCHEMBL573514 0.74
SCHEMBL29214271 0.73 HSD11B1 (0.41) HSD11B1MAOAMAOBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed
US-7935824-B2 Ethylenediamine derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2011-05-03 US disclosed