SCHEMBL7408342

SCHEMBL7408342

N[C@@H](CCc1c(O)noc1-c1ccc2ccccc2c1)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A11 Q9UPY5 1/20 0.45
SLC1A3 P43003 1/20 0.44
SLC1A2 P43004 1/20 0.44
SLC1A1 P43005 1/20 0.44
S1PR4 O95977 3/20 0.42
S1PR5 Q9H228 3/20 0.42
TPH1 P17752 5/20 0.37
KIF11 P52732 1/20 0.37
GRIK1 P39086 1/20 0.36
GRIK2 Q13002 1/20 0.36
GRIK3 Q13003 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ACMSD Q8TDX5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7408347 1.00 SLC7A11 (0.45) SLC7A11SLC1A3SLC1A2SLC1A1S1PR4
SCHEMBL8134760 0.88 SLC7A11 (0.52) SLC7A11SLC1A3SLC1A2SLC1A1S1PR4
SCHEMBL8134763 0.88 SLC7A11 (0.52) SLC7A11SLC1A3SLC1A2SLC1A1S1PR4
SCHEMBL8128585 0.87 KIF11 (0.39) SLC7A11KIF11MEN1CYP1A2KMT2A
SCHEMBL8128581 0.87 KIF11 (0.39) SLC7A11KIF11MEN1CYP1A2KMT2A
SCHEMBL7406145 0.81 TPH1 (0.46) TPH1KIF11GRIK1GRIK2KDM4E
SCHEMBL7406141 0.81 TPH1 (0.46) TPH1KIF11GRIK1GRIK2KDM4E
SCHEMBL8125246 0.80 NOS1 (0.43) KIF11GRIK1KMT2A
SCHEMBL8125242 0.80 NOS1 (0.43) KIF11GRIK1KMT2A
SCHEMBL7452720 0.78 SLC1A3 (0.35) SLC1A3SLC1A2SLC1A1GRIK1GRIK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994107-A1 5-Arylisoxazol-4-yl-substituted 2-amino carboxylic acid compounds H. LUNDBECK A/S (DK) 2000-04-19 EP disclosed
EP-0726896-A1 5-ARYLISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1996-08-21 EP disclosed
WO-1995012587-A1 5-ARYLISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1995-05-11 WO disclosed