SCHEMBL7410593

SCHEMBL7410593

Cc1ccc(S(=O)(=O)OC2CCc3c(c4cc(Cl)cc(C(F)(F)F)c4n3CCN3CCCC3)C2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 0.37
CYP2D6 P10635 2/20 0.36
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32
DRD3 P35462 1/20 0.32
MBTD1 Q05BQ5 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CYP1A2 P05177 1/20 0.31
CCR2 P41597 2/20 0.31
MAPK1 P28482 1/20 0.30
FPR2 P25090 1/20 0.30
PROKR1 Q8TCW9 1/20 0.30
SLC9A3 P48764 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410311 0.76 DRD2 (0.38) DRD2DRD3
SCHEMBL7405699 0.70 HTR6 (0.38) HTR6CYP2D6MEN1KMT2AALDH1A1
SCHEMBL7405351 0.69 PTGDR2 (0.43) CYP2D6L3MBTL1MEN1KMT2AALDH1A1
SCHEMBL7402689 0.69 DRD3 (0.39) HTR6DRD2DRD3
SCHEMBL7414266 0.69 PTGS1 (0.46) HTR6
SCHEMBL7406680 0.67 HTR6 (0.46) HTR6CYP2D6DRD1DRD3CYP1A2
SCHEMBL7463173 0.67 CGAS (0.38) HTR6CYP2D6CYP1A2
SCHEMBL7414173 0.66 HTR6 (0.50) HTR6CYP2D6DRD2DRD1DRD4
SCHEMBL7407904 0.66 HTR6 (0.51) HTR6CYP2D6CYP1A2MAPK1MEN1
SCHEMBL7410960 0.66 SIGMAR1 (0.37) CYP2D6DRD4MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4257952-A PSYCHOTROPIC DRUGS, ANALGESICS, ANTIHISTAMINES STERLING DRUG INC. (US) 1981-03-24 US disclosed
US-4172834-A ANALGESICS, ANTIHISTAMINES AND PSYCHOTROPIC AGENTS STERLING DRUG INC. (US) 1979-10-30 US disclosed
US-4062864-A ANALGESIC, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1977-12-13 US disclosed
US-3959309-A ANALGESICS, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1976-05-25 US disclosed