SCHEMBL7405351

SCHEMBL7405351

CC(=O)Nc1ccc2c(c1)c1c(n2CCN2CCN(C)CC2)CCC(OS(=O)(=O)c2ccc(C)cc2)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 6/20 0.43
CYP2D6 P10635 1/20 0.41
HTT P42858 2/20 0.39
MEN1 O00255 2/20 0.39
USP2 O75604 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 2/20 0.39
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
HTR1A P08908 2/20 0.37
KCNH2 Q12809 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
HTR1F P30939 1/20 0.37
ALDH1A1 P00352 4/20 0.37
LMNA P02545 2/20 0.37
KDM4E B2RXH2 1/20 0.36
ALOX15 P16050 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7413051 0.81 DRD2 (0.46) PTGDR2HTR1AHTR1DHTR1BHTR1F
SCHEMBL7405699 0.75 HTR6 (0.38) PTGDR2CYP2D6MEN1KMT2APOLB
SCHEMBL7412457 0.72 KMT2A (0.42) MEN1KMT2AMAPTSMN1; SMN2ALDH1A1
SCHEMBL7414173 0.70 HTR6 (0.50) PTGDR2CYP2D6HTR1AKCNH2
SCHEMBL7409122 0.70 PTGDR2 (0.44) PTGDR2CYP2D6
SCHEMBL7408736 0.69 HTR6 (0.52) PTGDR2CYP2D6HTR1AKCNH2
SCHEMBL7410593 0.69 HTR6 (0.37) CYP2D6MEN1KMT2AL3MBTL1ALDH1A1
SCHEMBL7403808 0.68 HTR6 (0.45)
SCHEMBL7406680 0.68 HTR6 (0.46) PTGDR2CYP2D6MEN1KMT2AHTR1A
SCHEMBL7407904 0.67 HTR6 (0.51) CYP2D6MEN1KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4257952-A PSYCHOTROPIC DRUGS, ANALGESICS, ANTIHISTAMINES STERLING DRUG INC. (US) 1981-03-24 US disclosed
US-4172834-A ANALGESICS, ANTIHISTAMINES AND PSYCHOTROPIC AGENTS STERLING DRUG INC. (US) 1979-10-30 US disclosed
US-4062864-A ANALGESIC, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1977-12-13 US disclosed
US-3959309-A ANALGESICS, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1976-05-25 US disclosed