SCHEMBL7410694

SCHEMBL7410694

Cc1ccc(-c2cccc3c4c([nH]c23)CCC(OS(=O)(=O)c2ccccc2)C4)cc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.37
CYP19A1 P11511 1/20 0.35
MCL1 Q07820 1/20 0.35
CYP2D6 P10635 2/20 0.34
PARP14 Q460N5 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
CYP1A2 P05177 1/20 0.33
NR2E1 Q9Y466 1/20 0.33
PTGS2 P35354 2/20 0.32
TP53 P04637 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
VDR P11473 1/20 0.31
RB1 P06400 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415797 0.85 CYP2D6 (0.40) HTR6CYP19A1CYP2D6CYP3A4CYP2C19
SCHEMBL7413413 0.81 MCL1 (0.39) MCL1PARP14
SCHEMBL7403630 0.81 CYP19A1 (0.50) HTR6CYP19A1CYP2D6CYP2C19CYP1A2
SCHEMBL7410972 0.75 TRPV1 (0.38) MCL1PARP14NR2E1HSD17B10RB1
SCHEMBL7414043 0.75 HTR6 (0.47) HTR6TP53RB1
SCHEMBL7463173 0.74 CGAS (0.38) HTR6CYP2D6CYP1A2PTGS2TP53
SCHEMBL7413193 0.73 HTR1A (0.44) HTR6
SCHEMBL7412807 0.73 CHRNA7 (0.41) PARP14NR2E1
SCHEMBL7407214 0.71 MAPT (0.40) HTR6CYP19A1CYP2D6TP53HPGD
SCHEMBL7410787 0.71 HTR2A (0.47) HTR6TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4257952-A PSYCHOTROPIC DRUGS, ANALGESICS, ANTIHISTAMINES STERLING DRUG INC. (US) 1981-03-24 US disclosed
US-4172834-A ANALGESICS, ANTIHISTAMINES AND PSYCHOTROPIC AGENTS STERLING DRUG INC. (US) 1979-10-30 US disclosed
US-4062864-A ANALGESIC, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1977-12-13 US disclosed
US-3959309-A ANALGESICS, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1976-05-25 US disclosed