SCHEMBL7412871

SCHEMBL7412871

Cc1cc(Br)ccc1S(=O)(=O)N[C@@H](Cc1ccc(OCCCONC(=N)N)cc1)C(=O)OC(=O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ITGB3 P05106 10/20 0.37
ITGA2B P08514 10/20 0.37
POLB P06746 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
TP53 P04637 1/20 0.33
F2 P00734 3/20 0.32
TMPRSS6 Q8IU80 3/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417980 0.92 MEN1 (0.40) MEN1KMT2AITGB3ITGA2BPOLB
Trifluoroacetic Acid SCHEMBL7412868 0.90 ITGB3 (0.47) MEN1KMT2AITGB3ITGA2BITGB1
SCHEMBL7414783 0.89 CYP3A4 (0.43) MEN1KMT2AITGB3ITGA2BPOLB
SCHEMBL7416202 0.89 MEN1 (0.38) MEN1KMT2AITGB3ITGA2BPOLB
SCHEMBL7415446 0.89 ITGB3 (0.39) MEN1KMT2AITGB3ITGA2BPOLB
SCHEMBL7408394 0.88 ITGB3 (0.37) ITGB3ITGA2BF2TMPRSS6CYP3A4
SCHEMBL7410416 0.88 L3MBTL1 (0.41) KMT2AITGB3ITGA2BF2TMPRSS6
SCHEMBL7412629 0.87 CTSL (0.43) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7414225 0.87 ITGB3 (0.50) MEN1KMT2AITGB3ITGA2BPOLB
SCHEMBL7418586 0.87 CYP3A4 (0.41) ITGB3ITGA2BF2TMPRSS6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed