SCHEMBL7416202

SCHEMBL7416202

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2ccc(Br)cc2OC(F)(F)F)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ITGB3 P05106 7/20 0.35
ITGA2B P08514 7/20 0.35
PTPN1 P18031 1/20 0.34
ALPL P05186 2/20 0.34
HSD17B1 P14061 5/20 0.34
HSD17B2 P37059 5/20 0.34
ADAMTS4 O75173 1/20 0.33
POLB P06746 1/20 0.33
PPARG P37231 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7416198 0.90 ITGB3 (0.43) MEN1KMT2AITGB3ITGA2BPPARG
SCHEMBL7471115 0.90 ITGB3 (0.44) MEN1KMT2AITGB3ITGA2BADAMTS4
SCHEMBL7412871 0.89 MEN1 (0.40) MEN1KMT2AITGB3ITGA2BPOLB
SCHEMBL7417980 0.89 MEN1 (0.40) MEN1KMT2AITGB3ITGA2BPTPN1
SCHEMBL7414783 0.88 CYP3A4 (0.43) MEN1KMT2AITGB3ITGA2BALPL
SCHEMBL7412629 0.86 CTSL (0.43) ITGB3ITGA2B
SCHEMBL7419584 0.85 F2 (0.42) MEN1KMT2AITGB3ITGA2BPTPN1
SCHEMBL7414402 0.84 POLB (0.49) MEN1KMT2AITGB3ITGA2BPOLB
SCHEMBL7410463 0.84 ITGB3 (0.38) MEN1KMT2AITGB3ITGA2BPOLB
SCHEMBL7415207 0.83 ITGB3 (0.50) ITGB3ITGA2BPPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed