SCHEMBL7413642

SCHEMBL7413642

CC(C)C(=O)c1nccn1COCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
OPRD1 P41143 3/20 0.39
OPRK1 P41145 2/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
TSHR P16473 2/20 0.38
MAPK1 P28482 2/20 0.38
HTT P42858 2/20 0.38
HPGD P15428 1/20 0.38
KDM4E B2RXH2 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
MAPT P10636 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3303697 0.87 CTSL (0.43) CTSLCTSSCTSKOPRD1SMN1; SMN2
SCHEMBL532075 0.85 KMT2A (0.38) CTSLCTSSCTSKSMN1; SMN2NPC1
SCHEMBL10242213 0.84 ATM (0.46) CTSLCTSSCTSKNPC1RAB9A
SCHEMBL27684880 0.82 CYP19A1 (0.41) OPRK1L3MBTL1
SCHEMBL7408571 0.75 MAPT (0.45) SMN1; SMN2ALDH1A1LMNATSHRMAPK1
SCHEMBL10434937 0.75 TSHR (0.44) CTSLCTSSCTSKALDH1A1LMNA
SCHEMBL9271702 0.74 MAPT (0.37) CTSLCTSSCTSKALDH1A1LMNA
SCHEMBL6579557 0.73 RAB9A (0.39) OPRD1OPRK1SMN1; SMN2NPC1RAB9A
SCHEMBL7357006 0.73 MAPT (0.40) SMN1; SMN2LMNATSHRMAPTTDP1
SCHEMBL26196832 0.73 MAOB (0.40) SMN1; SMN2NPC1RAB9AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5733882-A Retroviral protease inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1998-03-31 US disclosed
EP-0602069-A4 RETROVIRAL PROTEASE INHIBITORS. SMITHKLINE BEECHAM CORP (US) 1995-05-03 EP disclosed
EP-0602069-A1 RETROVIRAL PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1994-06-22 EP disclosed
WO-1993002057-A1 RETROVIRAL PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1993-02-04 WO disclosed