SCHEMBL7413755

SCHEMBL7413755

CC(C)Cn1nnnc1-c1ccc2c(c1)nc(COc1ccc(C#N)cc1)n2C

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.47
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
HDAC6 Q9UBN7 1/20 0.39
MAPT P10636 3/20 0.37
KDM4E B2RXH2 1/20 0.37
HIF1A Q16665 1/20 0.37
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
BRD4 O60885 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415639 0.85 F2 (0.49) PPARGNPC1RAB9AHDAC6
SCHEMBL7968222 0.79 ALDH1A1 (0.38) MAPTKDM4EBRD4ALDH1A1
Hydrochloric Acid SCHEMBL8028429 0.70 F2 (0.47)
SCHEMBL7377767 0.70 ALDH1A1 (0.53) PPARGNPC1RAB9AMAPTSMN1; SMN2
SCHEMBL7383468 0.69 RAB9A (0.58) PPARGNPC1RAB9AHDAC6MAPT
SCHEMBL6778595 0.67 PPARG (0.52) PPARGNPC1RAB9AALDH1A1CYP19A1
SCHEMBL7378592 0.65 PPARG (0.51) PPARGNPC1RAB9AHDAC6MAPT
SCHEMBL6781977 0.64 BRPF1 (0.48) PPARGNPC1RAB9AHDAC6MAPT
SCHEMBL6776552 0.64 PPARG (0.48) PPARGNPC1RAB9AHDAC6SMN1; SMN2
SCHEMBL7379857 0.62 HDAC6 (0.44) PPARGNPC1RAB9AHDAC6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000050419-A1 SUBSTITUTED BICYCLIC HETEROCYCLES AND THE USE THEREOF AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-08-31 WO disclosed