SCHEMBL7414006

SCHEMBL7414006

CC(C)(C)OC(=O)NC(C(N)=O)C(=O)N(CCNc1ccccc1)CCNc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.40
CTSS P25774 4/20 0.39
CTSK P43235 4/20 0.39
ATM Q13315 1/20 0.39
JAK3 P52333 1/20 0.38
BTK Q06187 1/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
REN P00797 3/20 0.38
PPARA Q07869 2/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
PPARG P37231 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
APP P05067 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417898 0.83 CTSK (0.47) BACE1CTSSCTSKATMCTSL
SCHEMBL7102658 0.76 CTSK (0.49) CTSSCTSKATMCTSLCTSB
SCHEMBL7419681 0.74 PPARG (0.44) CTSKPPARAALDH1A1PPARG
SCHEMBL7203913 0.70 MALT1 (0.59) CTSK
SCHEMBL13258281 0.70 ATM (0.50) CTSSCTSKATMCTSLCTSB
SCHEMBL13257888 0.70 ATM (0.50) CTSSCTSKATMCTSLCTSB
SCHEMBL13257955 0.70 ATM (0.50) CTSSCTSKATMCTSLCTSB
SCHEMBL12311224 0.70 GBA1 (0.44) CTSSCTSLCTSBALDH1A1HDAC1
SCHEMBL9186325 0.69 CA14 (0.55) BACE1RENALDH1A1HDAC1
SCHEMBL10126784 0.68 MEN1 (0.53) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140818-A1 AMIDOMALONAMIDES AND THEIR USE AS INHIBITORS OF MATRIX METALLOPROTEINASE Aventis Pharmaceuticals Inc. (US) 2001-10-10 EP disclosed
WO-2000040552-A1 AMIDOMALONAMIDES AND THEIR USE AS INHIBITORS OF MATRIX METALLOPROTEINASE AVENTIS PHARMACEUTICALS INC. (US) 2000-07-13 WO disclosed