SCHEMBL7414092

SCHEMBL7414092

COc1ccc(OC(C(=O)OCc2ccccc2)[C@@H]2CCN2)cn1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
PABPC1 P11940 1/20 0.45
ACACB O00763 5/20 0.37
ACACA Q13085 4/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TSHR P16473 1/20 0.36
CHRNA7 P36544 2/20 0.36
P4HTM Q9NXG6 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
HTR2C P28335 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414311 1.00 MEN1 (0.45) MEN1KMT2APABPC1ACACBACACA
SCHEMBL7411933 0.85 CYP3A4 (0.38) CYP3A4CYP2C9CYP2C19TSHRP4HTM
SCHEMBL7414234 0.85 CYP3A4 (0.38) CYP3A4CYP2C9CYP2C19TSHRP4HTM
SCHEMBL7410510 0.80 TSHR (0.35) CYP3A4CYP2C9CYP2C19TSHRP4HTM
SCHEMBL7414435 0.80 TSHR (0.35) CYP3A4CYP2C9CYP2C19TSHRP4HTM
SCHEMBL7414580 0.79 TSHR (0.35) MEN1KMT2ACYP3A4CYP2C9CYP2C19
SCHEMBL7415007 0.73 GLA (0.40) KMT2ACYP3A4CYP2C9CYP2C19TSHR
SCHEMBL6597590 0.73 HTR2C (0.41) CYP3A4CYP2C9CYP2C19TSHRHTR2C
SCHEMBL7414013 0.72 CHRNB2 (0.40) CHRNB2CHRNA4
SCHEMBL7411868 0.71 GLA (0.36) CYP3A4CYP2C9CYP2C19TSHRHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047690-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-11-02 EP disclosed
WO-1999032480-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1999-07-01 WO disclosed