SCHEMBL7414435

SCHEMBL7414435

Cc1cc(OC(C(=O)OCc2ccccc2)[C@H]2CCN2)cnc1F

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
P4HTM Q9NXG6 1/20 0.35
HTR2C P28335 1/20 0.35
SLC6A2 P23975 3/20 0.35
SLC6A3 Q01959 3/20 0.35
SLC6A4 P31645 2/20 0.35
LMNA P02545 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
S1PR1 P21453 1/20 0.34
S1PR5 Q9H228 1/20 0.34
PKM P14618 1/20 0.34
TP53 P04637 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
GLA P06280 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410510 1.00 TSHR (0.35) TSHRP4HTMHTR2CSLC6A2SLC6A3
SCHEMBL7414580 0.89 TSHR (0.35) TSHRHTR2CSLC6A2SLC6A3SLC6A4
SCHEMBL7411933 0.84 CYP3A4 (0.38) TSHRP4HTMHTR2CLMNAL3MBTL1
SCHEMBL7414234 0.84 CYP3A4 (0.38) TSHRP4HTMHTR2CLMNAL3MBTL1
SCHEMBL7414311 0.80 MEN1 (0.45) TSHRP4HTMHTR2CCYP3A4CYP2C9
SCHEMBL7414092 0.80 MEN1 (0.45) TSHRP4HTMHTR2CCYP3A4CYP2C9
SCHEMBL7405289 0.78 GLA (0.36) TSHRHTR2CSLC6A2SLC6A3SLC6A4
SCHEMBL7411868 0.78 GLA (0.36) TSHRHTR2CSLC6A2SLC6A3SLC6A4
SCHEMBL7415007 0.78 GLA (0.40) TSHRSLC6A2SLC6A3SLC6A4L3MBTL1
SCHEMBL7476578 0.76 ALKBH1 (0.36) P4HTMLMNAL3MBTL1S1PR1S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047690-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-11-02 EP disclosed
WO-1999032480-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1999-07-01 WO disclosed