SCHEMBL7414402

SCHEMBL7414402

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2ccccc2Br)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.49
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ITGB3 P05106 8/20 0.38
ITGA2B P08514 8/20 0.38
RECQL P46063 1/20 0.38
F2 P00734 6/20 0.37
TMPRSS6 Q8IU80 4/20 0.37
PRSS1 P07477 1/20 0.34
PRSS2 P07478 1/20 0.34
PRSS3 P35030 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414101 0.91 ITGB3 (0.40) POLBITGB3ITGA2BF2TMPRSS6
SCHEMBL7413080 0.90 MMP7 (0.40) POLBMEN1KMT2AITGB3ITGA2B
SCHEMBL7415119 0.90 ITGB1 (0.39) POLBITGB3ITGA2BF2TMPRSS6
SCHEMBL7415446 0.90 ITGB3 (0.39) POLBMEN1KMT2AITGB3ITGA2B
SCHEMBL7694227 0.89 F10 (0.41) ITGB3ITGA2BF2TMPRSS6
Trifluoroacetic Acid SCHEMBL7414396 0.89 POLB (0.49) POLBITGB3ITGA2BF2TMPRSS6
SCHEMBL7417592 0.88 ITGB3 (0.49) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7410463 0.88 ITGB3 (0.38) POLBMEN1KMT2AITGB3ITGA2B
SCHEMBL7415626 0.88 HRH2 (0.37) POLBITGB3ITGA2BF2TMPRSS6
SCHEMBL7415041 0.87 AR (0.38) POLBMEN1KMT2AITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed