SCHEMBL7414115

SCHEMBL7414115

CN1CCN(C(=O)c2ccc3c(c2)N=C(N)c2sccc2C3)CC1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
HPGD P15428 4/20 0.43
TSHR P16473 1/20 0.43
POLB P06746 3/20 0.41
HRH4 Q9H3N8 2/20 0.41
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
ALOX15 P16050 1/20 0.40
CTSD P07339 2/20 0.39
KCNH2 Q12809 1/20 0.39
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417430 0.92 CTSD (0.47) KMT2AMEN1HPGDPOLBALDH1A1
SCHEMBL7592584 0.91 KMT2A (0.44) KMT2AMEN1HPGDTSHRPOLB
SCHEMBL7402968 0.88 HSP90AA1 (0.40) KMT2AALDH1A1MAPTCTSD
SCHEMBL7380703 0.82 NOS3 (0.37) KMT2AMEN1TSHRALDH1A1MAPT
SCHEMBL7375377 0.74 NOS2 (0.42) KMT2AMEN1HPGDALDH1A1MAPT
SCHEMBL7423582 0.71 NOS2 (0.41)
SCHEMBL7386220 0.70 AOC3 (0.37) KMT2AMEN1HPGDALDH1A1MAPT
SCHEMBL7423018 0.69 NOS3 (0.40) TSHRPOLBALDH1A1
SCHEMBL7417662 0.69 NOS2 (0.41)
SCHEMBL7563046 0.68 NOS2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000073313-A1 NEW TRICYCLIC AMIDINE DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2000-12-07 WO claimed
WO-2000073313-A1 NEW TRICYCLIC AMIDINE DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2000-12-07 WO disclosed