SCHEMBL7417430

SCHEMBL7417430

NC1=Nc2cc(C(=O)N3CCCC3)ccc2Cc2ccsc21

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSD P07339 2/20 0.47
NPC1 O15118 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
POLB P06746 1/20 0.39
HPGD P15428 5/20 0.39
ADORA2A P29274 2/20 0.39
ALDH1A1 P00352 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HSD11B1 P28845 1/20 0.39
KDM1A O60341 1/20 0.38
GRIA3 P42263 1/20 0.38
GRIA4 P48058 1/20 0.38
L3MBTL3 Q96JM7 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414115 0.92 KMT2A (0.44) CTSDTLR8TLR7MEN1KMT2A
SCHEMBL7402968 0.89 HSP90AA1 (0.40) CTSDNPC1KMT2AALDH1A1L3MBTL3
SCHEMBL7592584 0.83 KMT2A (0.44) MEN1KMT2APOLBHPGDADORA2A
SCHEMBL7380703 0.83 NOS3 (0.37) NPC1MEN1KMT2AALDH1A1KDM4E
SCHEMBL7375377 0.75 NOS2 (0.42) NPC1MEN1KMT2AHPGDALDH1A1
SCHEMBL7423018 0.72 NOS3 (0.40) NPC1POLBALDH1A1
SCHEMBL7423582 0.72 NOS2 (0.41)
SCHEMBL7417662 0.69 NOS2 (0.41)
SCHEMBL7396252 0.69 ALDH1A1 (0.37) ALDH1A1
SCHEMBL7386220 0.69 AOC3 (0.37) TLR7MEN1KMT2AHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000073313-A1 NEW TRICYCLIC AMIDINE DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2000-12-07 WO disclosed