SCHEMBL7414356

SCHEMBL7414356

NN=Cc1ccc(CCCCNC(=O)[C@H](CC(=O)O)NC(=O)OCc2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 8/20 0.52
CA5A P35218 1/20 0.50
CA2 P00918 1/20 0.49
CA1 P00915 1/20 0.48
TPSAB1 Q15661 1/20 0.47
HTT P42858 1/20 0.47
FOLH1 Q04609 1/20 0.46
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
CAPN1 P07384 1/20 0.46
CAPN2 P17655 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.46
SIRT1 Q96EB6 1/20 0.46
SIRT3 Q9NTG7 1/20 0.46
PTGER4 P35408 1/20 0.46
CA4 P22748 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417109 1.00 CASP1 (0.52) CASP1CA5ACA2CA1TPSAB1
SCHEMBL8995553 0.93 FOLH1 (0.52) CA5ACA2CA1TPSAB1FOLH1
SCHEMBL7415259 0.93 FOLH1 (0.52) CA5ACA2CA1TPSAB1FOLH1
SCHEMBL7417452 0.90 CA1 (0.51) CA5ACA2CA1TPSAB1FOLH1
SCHEMBL8995555 0.86 MEN1 (0.55) CA5ACA1TPSAB1CAPN1CAPN2
SCHEMBL7471588 0.84 FOLH1 (0.52) TPSAB1FOLH1ITGB3CAPN1CAPN2
SCHEMBL7414342 0.83 CASP1 (0.53) CASP1CA5ACA2CA1TPSAB1
SCHEMBL7414413 0.83 CASP1 (0.53) CASP1CA5ACA2CA1TPSAB1
SCHEMBL7414348 0.83 CASP1 (0.53) CASP1CA5ACA2CA1TPSAB1
SCHEMBL8995559 0.77 KMT2A (0.44) CASP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552431-A ANTICOAGULANTS G. D. SEARLE & CO. (US) 1996-09-03 US disclosed
US-5424334-A Peptide mimetic compounds useful as platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1995-06-13 US disclosed
WO-1993012074-A1 PEPTIDE MIMETIC COMPOUNDS USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-06-24 WO disclosed