SCHEMBL7414938

SCHEMBL7414938

CC(C)[C@H](N)C(=O)N(C(=O)CCc1ccccc1)[C@@H](C)C(=O)NC(CC(=O)O)C(=O)C=[N+]=[N-]

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
MMP8 P22894 1/20 0.35
CASP1 P29466 7/20 0.34
LTA4H P09960 2/20 0.33
IL1B P01584 1/20 0.33
CASP3 P42574 3/20 0.33
CASP8 Q14790 2/20 0.33
CASP7 P55210 1/20 0.33
MME P08473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423470 0.88 F2 (0.41)
SCHEMBL7277260 0.86 CASP1 (0.41) KMT2AMEN1CASP1CASP3CASP8
SCHEMBL7286995 0.84 CASP1 (0.40) KMT2AMEN1CASP1CASP3CASP8
SCHEMBL7417508 0.84 CASP1 (0.35) CASP1CASP3CASP8CASP7
SCHEMBL7285059 0.83 CASP3 (0.44) CASP1CASP3CASP8CASP7
SCHEMBL7416641 0.81 CASP1 (0.34) MMP8CASP1CASP3CASP8CASP7
SCHEMBL7424734 0.81 ERAP2 (0.36) MMP8
SCHEMBL7277122 0.81 CASP1 (0.51) CASP1IL1B
SCHEMBL7277381 0.79 CASP1 (0.58) CASP1CASP3
SCHEMBL7301728 0.78 CTSC (0.47) KMT2AMEN1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014777-A1 PEPTIDYL DERIVATIVES AS INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME MERCK & CO., INC. (US) 1993-08-05 WO disclosed