SCHEMBL741499

SCHEMBL741499

COC(C#N)C(=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
TDP1 Q9NUW8 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 4/20 0.42
CYP3A4 P08684 1/20 0.42
LMNA P02545 4/20 0.41
CES2 O00748 2/20 0.41
CES1 P23141 2/20 0.41
HTT P42858 1/20 0.40
PGR P06401 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
HTR2A P28223 1/20 0.40
HRH1 P35367 1/20 0.40
KCNH2 Q12809 1/20 0.40
MDM2 Q00987 1/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11331689 0.82 SLC6A3 (0.40) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL25213754 0.82 HSD17B10 (0.47) L3MBTL1ALDH1A1CYP3A4LMNAHTT
SCHEMBL20075175 0.82 LMNA (0.47) TSHRTDP1ALDH1A1LMNACES2
SCHEMBL30737544 0.82 RAPGEF3 (0.44) TSHRL3MBTL1ALDH1A1LMNACES2
SCHEMBL21741440 0.82 GSK3B (0.56) ALDH1A1RAB9AKMT2AMAPTPOLB
SCHEMBL8315333 0.82 CES2 (0.57) TSHRALDH1A1CES2CES1NPC1
SCHEMBL741380 0.77 CES1 (0.40) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL28273393 0.76 CES2 (0.42) TDP1L3MBTL1ALDH1A1CYP3A4LMNA
SCHEMBL2989614 0.75 KMT2A (0.47) TSHRTDP1L3MBTL1ALDH1A1CYP3A4
SCHEMBL9018972 0.75 NPC1 (0.42) TSHRTDP1L3MBTL1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105272883-B A kind of preparation method of the fluoro benzoyl acetonitrile of high-purity 4 天津市科莱博瑞科技有限公司 2017-09-22 CN disclosed
CN-105272883-A Preparation method for high-purity 4-fluorobenzoylacetonitrile TIANJIN KELAI BORUI TECHNOLOGY CO LTD 2016-01-27 CN disclosed
EP-2430029-A1 THIENO [2, 3-B]PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS Katholieke Universiteit Leuven (BE) 2012-03-21 EP disclosed
WO-2010130842-A1 THIENO [2, 3-B] PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2010-11-18 WO disclosed
EP-0315698-B1 THIENO(TRIAZOLO)DIAZEPINE COMPOUNDS AND MEDICINAL APPLICATION OF THE SAME YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1993-03-03 EP disclosed
US-4960770-A Vasodilating agents, cardiovascular disorder YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1990-10-02 US disclosed
EP-0315698-A1 THIENO(TRIAZOLO)DIAZEPINE COMPOUNDS AND MEDICINAL APPLICATION OF THE SAME YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1989-05-17 EP disclosed