SCHEMBL7415419

SCHEMBL7415419

O=C(O)C1CN(c2ccccc2)C(=O)c2[nH]c3ccc(F)cc3c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 2/20 0.41
GLA P06280 1/20 0.41
HTT P42858 1/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
KCNH2 Q12809 1/20 0.40
MAPKAPK2 P49137 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
MPO P05164 1/20 0.38
XDH P47989 1/20 0.38
MAP2 P11137 1/20 0.38
CCNB2 O95067 1/20 0.38
CDK1 P06493 1/20 0.38
CCNB1 P14635 1/20 0.38
GSK3B P49841 1/20 0.38
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414405 0.87 KCNH2 (0.39) KDM4EALDH1A1GAAGLAHTT
SCHEMBL7410799 0.74 ROCK2 (0.42) ALDH1A1GAAMAPKAPK2LMNA
SCHEMBL8241808 0.74 CA1 (0.42) KDM4EALDH1A1GAAGLAHTT
SCHEMBL7406913 0.72 KDM4E (0.43) KDM4EALDH1A1GAAHTTHPGD
SCHEMBL9734334 0.68 NPC1 (0.42) ALDH1A1HPGD
SCHEMBL31530864 0.67 NOTUM (0.45) ALDH1A1HTTLMNA
SCHEMBL7414202 0.65 MEN1 (0.37)
Hydrochloric Acid SCHEMBL11259771 0.65 MAPKAPK2 (0.43) KDM4EALDH1A1HTR2AHTR2CKCNH2
SCHEMBL11256635 0.65 MAPKAPK2 (0.60) HTR2AHTR2CMAPKAPK2FEN1SIGMAR1
SCHEMBL6295699 0.63 KDM4E (0.59) KDM4EALDH1A1GAAGLAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6075021-A 1H-pyrido[3,4-b]indole-4-carboxamide derivatives, preparation and application thereof in therapeutics SYNTHELABO (FR) 2000-06-13 US disclosed