SCHEMBL7416029

SCHEMBL7416029

O=C(O)c1[nH]c(CBr)nc1Br

nearest known ligand 0.30

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.30
MAPK1 P28482 1/20 0.30
CASP1 P29466 1/20 0.30
CYP2C19 P33261 1/20 0.30
PIN1 Q13526 1/20 0.30
GPR35 Q9HC97 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23930862 0.80 PIN1 (0.44) CYP1A2MAPK1CASP1CYP2C19PIN1
SCHEMBL3032708 0.71 GPR35 (0.37) CYP1A2MAPK1CASP1CYP2C19PIN1
SCHEMBL6494249 0.64 HCAR2 (0.43) PIN1
SCHEMBL23930812 0.63 NPSR1 (0.45)
SCHEMBL24283838 0.63 LMNA (0.37) MAPK1
SCHEMBL2804373 0.60 PIN1 (0.44) CYP1A2MAPK1CASP1CYP2C19PIN1
SCHEMBL2778487 0.60 TP53 (0.44) PIN1
SCHEMBL11008167 0.60 PIN1 (0.44) CYP1A2MAPK1CASP1CYP2C19PIN1
SCHEMBL2522013 0.60 PIN1 (0.48) CYP1A2MAPK1CASP1CYP2C19PIN1
SCHEMBL2491316 0.59 KDM4E (0.41) CYP1A2CYP2C19PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994011398-A1 CYCLIC COMPOUNDS LINKED BY A HETEROCYCLIC RING USEFUL AS INHIBITORS OF PLATELET GLYCOPROTEIN IIb/IIIa THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-05-26 WO disclosed