SCHEMBL7416244

SCHEMBL7416244

N#CC1(N(Cc2cccnc2)C(=O)[CH]CC2(C(N)=O)CCCCC2)CCNC1

nearest known ligand 0.31

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPR132 Q9UNW8 1/20 0.31
PDE7B Q9NP56 1/20 0.31
ABL1 P00519 1/20 0.31
RIN1 Q13671 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
NAMPT P43490 1/20 0.31
RECQL P46063 1/20 0.30
ALDH1A1 P00352 2/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6371523 0.89 SNCA (0.33)
SCHEMBL7419503 0.84 HSD11B1 (0.32) ALDH1A1
SCHEMBL7420829 0.84 SNCA (0.34) ALDH1A1
SCHEMBL7422302 0.84 SLC6A2 (0.35)
SCHEMBL7014387 0.83 SNCA (0.33) ALDH1A1
SCHEMBL7418232 0.83 PTGES (0.35)
SCHEMBL7416951 0.82
SCHEMBL7411437 0.82 CTSB (0.31)
SCHEMBL7573990 0.82
SCHEMBL7414438 0.81 PTGES (0.36) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed