SCHEMBL7418232

SCHEMBL7418232

N#CC1(N(Cc2cccc(Oc3ccccc3)c2)C(=O)[CH]CC2(C(N)=O)CCCCC2)CCNC1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGES O14684 3/20 0.35
FFAR4 Q5NUL3 1/20 0.33
EGLN2 Q96KS0 3/20 0.33
EGLN1 Q9GZT9 3/20 0.33
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CHRM3 P20309 1/20 0.31
DAGLA Q9Y4D2 3/20 0.31
ALOX5 P09917 2/20 0.31
P2RX3 P56373 2/20 0.31
P2RX2 Q9UBL9 2/20 0.31
FAAH O00519 1/20 0.31
EPOR P19235 1/20 0.31
ABHD6 Q9BV23 1/20 0.30
FKBP1A P62942 1/20 0.30
HRH1 P35367 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414438 0.92 PTGES (0.36) PTGESEPOR
SCHEMBL6371523 0.91 SNCA (0.33)
SCHEMBL7422302 0.87 SLC6A2 (0.35)
SCHEMBL7420829 0.85 SNCA (0.34)
SCHEMBL7014387 0.84 SNCA (0.33) TSHR
SCHEMBL7411437 0.84 CTSB (0.31)
SCHEMBL7416244 0.83 GPR132 (0.31)
SCHEMBL7419503 0.82 HSD11B1 (0.32)
SCHEMBL7416951 0.82
SCHEMBL7573990 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed