SCHEMBL7420829

SCHEMBL7420829

N#CC1(N(Cc2ccccc2)C(=O)[CH]CC2(C(N)=O)CCCCC2)CCNCC1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SNCA P37840 2/20 0.34
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
CTSB P07858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6371523 0.94 SNCA (0.33) SNCACTSSCTSK
SCHEMBL7014387 0.91 SNCA (0.33) SNCACTSSCTSKALDH1A1MAPK1
SCHEMBL7419258 0.90 CTSB (0.32) CTSSCTSB
SCHEMBL7418232 0.85 PTGES (0.35)
SCHEMBL7419503 0.85 HSD11B1 (0.32) ALDH1A1
SCHEMBL7411437 0.85 CTSB (0.31) CTSSCTSB
SCHEMBL7422302 0.85 SLC6A2 (0.35)
SCHEMBL7414438 0.84 PTGES (0.36) ALDH1A1MAPK1
SCHEMBL7416244 0.84 GPR132 (0.31) ALDH1A1
SCHEMBL7416951 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed