SCHEMBL7417865

SCHEMBL7417865

Cc1ccccc1-n1c(=O)[nH]c(=O)c2ncn(Cc3ccccc3C(F)(F)F)c21

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
YTHDC1 Q96MU7 1/20 0.44
P2RX7 Q99572 2/20 0.39
CNR2 P34972 8/20 0.39
C5AR1 P21730 1/20 0.39
MAPK1 P28482 2/20 0.39
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
ATM Q13315 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PNP P00491 1/20 0.37
TRPC5 Q9UL62 1/20 0.37
CNR1 P21554 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416426 0.82 HPGD (0.49) MAPK1ALDH1A1TDP1KDM4EPNP
SCHEMBL7423403 0.74 KMT2A (0.48) ALDH1A1KDM4EPNP
SCHEMBL7417864 0.71 HCAR1 (0.42) P2RX7C5AR1ALDH1A1TDP1KDM4E
SCHEMBL7604062 0.67 PNP (0.53) MAPK1KDM4EPNP
SCHEMBL7417859 0.66 PDE4A (0.69) C5AR1
SCHEMBL7467503 0.64 C5AR1 (0.49) P2RX7C5AR1ALDH1A1TDP1KDM4E
SCHEMBL7421519 0.63 PNP (0.49) MAPK1PNPCNR1
SCHEMBL17931795 0.63 L3MBTL1 (0.51) P2RX7C5AR1ALDH1A1TDP1KDM4E
SCHEMBL16053109 0.63 ALDH1A1 (0.68) MAPK1ALDH1A1TDP1GAA
SCHEMBL27501339 0.62 BRD4 (0.58) KDM4ENPSR1PNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821366-A Xanthines and their therapeutic use CHIROSCIENCE LIMITED (GB) 1998-10-13 US claimed
EP-0825993-A1 XANTHINES AND THEIR THERAPEUTIC USE Chiroscience Limited (GB) 1998-03-04 EP claimed
WO-1996036638-A1 XANTHINES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO claimed
EP-0825993-A1 XANTHINES AND THEIR THERAPEUTIC USE Chiroscience Limited (GB) 1998-03-04 EP disclosed
WO-1996036638-A1 XANTHINES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO disclosed