SCHEMBL7416426

SCHEMBL7416426

Cc1ccccc1-n1c(=O)[nH]c(=O)c2ncn(Cc3ccccc3)c21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.49
PNP P00491 1/20 0.48
BRD4 O60885 1/20 0.47
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
LMNA P02545 2/20 0.43
KDM4E B2RXH2 2/20 0.43
POLB P06746 2/20 0.43
MAPK1 P28482 1/20 0.43
PARN O95453 1/20 0.43
CNOT7 Q9UIV1 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7604062 0.84 PNP (0.53) HPGDPNPBRD4PDE4ALMNA
SCHEMBL7417865 0.82 YTHDC1 (0.44) PNPKDM4EMAPK1ALDH1A1TDP1
SCHEMBL7421519 0.80 PNP (0.49) HPGDPNPBRD4PDE4AMAPK1
SCHEMBL27501339 0.79 BRD4 (0.58) HPGDPNPBRD4KDM4EPARN
SCHEMBL7421933 0.78 PNP (0.47) HPGDPNPBRD4PDE4APDE4B
SCHEMBL3110932 0.76 PDE1A (0.53) HPGDPNPBRD4PARNCNOT7
SCHEMBL3115743 0.75 ALDH1A1 (0.51) HPGDPNPBRD4PDE4APDE4B
SCHEMBL7420637 0.73 PGR (0.43) HPGDPNPPDE4ALMNAKDM4E
SCHEMBL4624547 0.72 BRD4 (0.52) HPGDPNPBRD4KDM4EPOLB
SCHEMBL7423403 0.71 KMT2A (0.48) PNPPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825993-A1 XANTHINES AND THEIR THERAPEUTIC USE Chiroscience Limited (GB) 1998-03-04 EP claimed
WO-1996036638-A1 XANTHINES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO claimed