SCHEMBL7417997

SCHEMBL7417997

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)CCCCl)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 17/20 0.44
ITGA2B P08514 17/20 0.44
ITGAV P06756 1/20 0.40
CHRM2 P08172 1/20 0.40
SLC6A4 P31645 1/20 0.40
ITGB1 P05556 1/20 0.34
ITGA5 P08648 1/20 0.34
F2 P00734 2/20 0.33
TMPRSS6 Q8IU80 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7409569 0.92 ITGB3 (0.54) ITGB3ITGA2BITGAVCHRM2SLC6A4
Trifluoroacetic Acid SCHEMBL7417991 0.89 ITGB3 (0.55) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7415207 0.88 ITGB3 (0.50) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7414434 0.85 F2 (0.42) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7415975 0.85 ITGB3 (0.59) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7417592 0.85 ITGB3 (0.49) ITGB3ITGA2BITGAVF2TMPRSS6
SCHEMBL7416602 0.85 ITGB3 (0.38) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7415327 0.85 ITGB1 (0.42) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7415235 0.84 KCNA5 (0.44) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7417563 0.84 ITGB3 (0.39) ITGB3ITGA2BITGAVCHRM2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed