SCHEMBL7415207

SCHEMBL7415207

CS(=O)(=O)N[C@@H](Cc1ccc(OCCCONC(=N)N)cc1)C(=O)OC(=O)C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.50
ITGA2B P08514 13/20 0.50
PPARG P37231 3/20 0.39
F2 P00734 2/20 0.35
TMPRSS6 Q8IU80 2/20 0.35
ITGAV P06756 1/20 0.35
CHRM2 P08172 1/20 0.35
SLC6A4 P31645 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA9 Q16790 1/20 0.35
ACACB O00763 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415235 0.89 KCNA5 (0.44) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7417563 0.89 ITGB3 (0.39) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7415446 0.89 ITGB3 (0.39) ITGB3ITGA2BPPARGF2TMPRSS6
SCHEMBL7409569 0.89 ITGB3 (0.54) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7416574 0.89 ITGB3 (0.45) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7694791 0.89 MMP2 (0.45) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7417592 0.88 ITGB3 (0.49) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7414101 0.88 ITGB3 (0.40) ITGB3ITGA2BF2TMPRSS6
Trifluoroacetic Acid SCHEMBL7415198 0.88 ITGB3 (0.63) ITGB3ITGA2BPPARGITGAVCHRM2
SCHEMBL7417997 0.88 ITGB3 (0.44) ITGB3ITGA2BF2TMPRSS6ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed