SCHEMBL7422223

SCHEMBL7422223

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)C(F)(F)C(=O)NC(COCc1ccccc1)COCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.45
ITGA2B P08514 6/20 0.45
MME P08473 1/20 0.45
ACE P12821 1/20 0.45
CPA1 P15085 1/20 0.45
ACE2 Q9BYF1 1/20 0.45
CMA1 P23946 3/20 0.44
CTSD P07339 2/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
PTPN1 P18031 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
CASP3 P42574 1/20 0.42
CASP7 P55210 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7933938 0.93 CTSD (0.47) ITGB3ITGA2BMMEACECPA1
SCHEMBL8945566 0.93 CTSD (0.47) ITGB3ITGA2BMMEACECPA1
SCHEMBL8041651 0.89 MME (0.47) ITGB3ITGA2BMMEACECPA1
SCHEMBL8945610 0.88 MME (0.45) ITGB3ITGA2BMMEACECPA1
SCHEMBL8736216 0.88 CTSD (0.53) ITGB3ITGA2BMMEACECPA1
SCHEMBL7418725 0.87 MME (0.46) MMEACECPA1ACE2
SCHEMBL7417968 0.87 GPR132 (0.44) CTSDCTSSCTSK
SCHEMBL7421246 0.87 GPR132 (0.44) CTSDCTSSCTSK
SCHEMBL7422846 0.86 CTSD (0.44) ITGB3ITGA2BMMEACECPA1
SCHEMBL7416869 0.86 MME (0.43) ITGB3ITGA2BMMEACECPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995001958-A1 DIFLUORO STATONE ANALOGS MERRELL PHARMACEUTICALS INC. (US) 1995-01-19 WO claimed
US-6114380-A ANTIVIRAL AGENT; ADMINISTERING TO TREAT HIV INFECTION; N-(4-(N-BENZYLOXYCARBONYL-L-VALYL)AMINO-2,2-DIFLUORO-1,3-DIOXO-5-(4-(2-N -MORPHOLYL)ETHYLOXY)PHENYL-PENTYL)-O-((2-PYRIDYL)METHYL)-D-VALINOL, FOR EXAMPLE MERRELL PHARMACEUTICALS INC. (US) 2000-09-05 US disclosed
WO-1995001958-A1 DIFLUORO STATONE ANALOGS MERRELL PHARMACEUTICALS INC. (US) 1995-01-19 WO disclosed