SCHEMBL7416869

SCHEMBL7416869

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)C(F)(F)C(=O)NC(c1ccccn1)c1ccccn1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MME P08473 1/20 0.43
ACE P12821 1/20 0.43
CPA1 P15085 1/20 0.43
ACE2 Q9BYF1 1/20 0.43
REN P00797 1/20 0.43
ITGB3 P05106 2/20 0.43
ITGA2B P08514 2/20 0.43
CTSD P07339 2/20 0.43
CTSS P25774 4/20 0.43
CTSL P07711 3/20 0.43
CTSK P43235 2/20 0.43
CTSB P07858 2/20 0.42
CMA1 P23946 1/20 0.42
CASP3 P42574 2/20 0.41
CASP7 P55210 2/20 0.41
HDAC8 Q9BY41 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8041651 0.90 MME (0.47) MMEACECPA1ACE2ITGB3
SCHEMBL8945610 0.86 MME (0.45) MMEACECPA1ACE2ITGB3
SCHEMBL8736216 0.86 CTSD (0.53) MMEACECPA1ACE2ITGB3
SCHEMBL8945318 0.86 CTSD (0.46) MMEACECPA1ACE2ITGB3
SCHEMBL7422223 0.86 ITGB3 (0.45) MMEACECPA1ACE2ITGB3
SCHEMBL8364492 0.85 CTSD (0.48) RENCTSDCMA1CASP3CASP7
SCHEMBL8041703 0.85 CTSD (0.49) RENITGB3ITGA2BCTSDCTSS
SCHEMBL7933938 0.85 CTSD (0.47) MMEACECPA1ACE2REN
SCHEMBL8945566 0.85 CTSD (0.47) MMEACECPA1ACE2REN
SCHEMBL7423864 0.85 REN (0.45) MMEACECPA1ACE2REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0707564-B1 DIFLUORO STATONE ANALOGS MERRELL PHARMA INC (US) 2000-09-20 EP claimed
WO-1995001958-A1 DIFLUORO STATONE ANALOGS MERRELL PHARMACEUTICALS INC. (US) 1995-01-19 WO claimed
EP-0707564-B1 DIFLUORO STATONE ANALOGS MERRELL PHARMA INC (US) 2000-09-20 EP disclosed
US-6114380-A ANTIVIRAL AGENT; ADMINISTERING TO TREAT HIV INFECTION; N-(4-(N-BENZYLOXYCARBONYL-L-VALYL)AMINO-2,2-DIFLUORO-1,3-DIOXO-5-(4-(2-N -MORPHOLYL)ETHYLOXY)PHENYL-PENTYL)-O-((2-PYRIDYL)METHYL)-D-VALINOL, FOR EXAMPLE MERRELL PHARMACEUTICALS INC. (US) 2000-09-05 US disclosed
WO-1995001958-A1 DIFLUORO STATONE ANALOGS MERRELL PHARMACEUTICALS INC. (US) 1995-01-19 WO disclosed