SCHEMBL7422899

SCHEMBL7422899

CC(C)(C)OC(=O)N[C@]1(C(N)c2ccc3ccncc3c2)CCNC1=O

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.34
ROCK2 O75116 7/20 0.33
AKT1 P31749 3/20 0.33
NAMPT P43490 4/20 0.32
PPIA P62937 2/20 0.32
NR3C1 P04150 1/20 0.31
ROCK1 Q13464 1/20 0.31
LATS1 O95835 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7369599 0.89 HPGDS (0.34) HPGDSROCK2AKT1NAMPTPPIA
SCHEMBL7373241 0.89 HPGDS (0.34) HPGDSROCK2AKT1NAMPTPPIA
SCHEMBL7374405 0.85 AKT1 (0.35) HPGDSROCK2AKT1NAMPTLATS1
SCHEMBL7369928 0.82 ROCK2 (0.41) ROCK2AKT1PPIA
SCHEMBL7373193 0.78 AKT1 (0.37) HPGDSROCK2AKT1NAMPTLATS1
Trifluoroacetic Acid SCHEMBL7376828 0.77 AKT1 (0.33) ROCK2AKT1ROCK1
Trifluoroacetic Acid SCHEMBL7384596 0.73 ROCK2 (0.36) HPGDSROCK2NAMPT
SCHEMBL7377427 0.72 HPGDS (0.31) HPGDS
SCHEMBL7367861 0.70 ROCK2 (0.40) ROCK2AKT1PPIA
SCHEMBL16246731 0.70 ROCK2 (0.44) ROCK2AKT1NR3C1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0975600-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS ANTITHROMBOTIC AGENTS Akzo Nobel N.V. (NL) 2000-02-02 EP disclosed
WO-1998047876-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS ANTITHROMBOTIC AGENTS AKZO NOBEL N.V. (NL) 1998-10-29 WO disclosed