SCHEMBL7423243

SCHEMBL7423243

C[Si](C)(C)OC1=Cc2ccccc2C1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.41
CYP11B2 P19099 3/20 0.38
CYP11B1 P15538 2/20 0.38
TRPA1 O75762 3/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
ACHE P22303 1/20 0.35
GPR84 Q9NQS5 1/20 0.34
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31
KDM4E B2RXH2 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CYP19A1 P11511 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9797964 0.83 CYP11B1 (0.39) PTGS2CYP11B2CYP11B1MAOBGPR84
SCHEMBL6907784 0.82 PTGS2 (0.37) PTGS2CYP11B2CYP11B1TRPA1MAOA
SCHEMBL12797023 0.80 TSHR (0.35) PTGS2CYP11B2CYP11B1MAOAMAOB
SCHEMBL7034657 0.80 PTGS2 (0.36) PTGS2CYP11B2CYP11B1TRPA1MAOA
SCHEMBL7031079 0.79 PTGS2 (0.35) PTGS2CYP11B2CYP11B1TRPA1MAOA
SCHEMBL8031056 0.78 PTGS2 (0.53) PTGS2CYP11B2CYP11B1TRPA1MAOA
SCHEMBL7196319 0.77 ACHE (0.35) PTGS2CYP11B2CYP11B1ACHE
SCHEMBL6908479 0.75 PTGS2 (0.33) PTGS2CYP11B2CYP11B1ACHE
SCHEMBL7202063 0.75 PTGS2 (0.35) PTGS2CYP11B2CYP11B1TRPA1MAOA
SCHEMBL6907494 0.74 PTGS2 (0.41) PTGS2CYP11B2CYP11B1TRPA1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214303-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001016121-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF MERCK & CO., INC. (US) 2001-03-08 WO disclosed
US-5366984-A Fungicides, insecticides BASF AKTIENGESELLSCHAFT (DE) 1994-11-22 US disclosed
US-5294628-A Fungicides, insecticides, pesticides BASF AKTIENGESELLSCHAFT (DE) 1994-03-15 US disclosed
EP-0378755-B1 Heterocyclically substituted alpha-aryl acryl acid methyl esters and their use BASF AG (DE) 1993-12-29 EP disclosed
US-5250553-A Fungicides; pesticides BASF AKTIENGESELLSCHAFT (DE) 1993-10-05 US disclosed
US-5166216-A Fungicides, pesticides, insecticides BASF AKTIENGESELLSCHAFT (DE) 1992-11-24 US disclosed