SCHEMBL7423402

SCHEMBL7423402

Nc1ccccc1-n1c(=O)[nH]c(=O)c2[nH]c(Cc3ccccc3F)nc21

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.46
PCK1 P35558 3/20 0.42
HCAR1 Q9BXC0 2/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 1/20 0.37
DAO P14920 1/20 0.36
HPGD P15428 1/20 0.36
PNP P00491 1/20 0.36
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
USP2 O75604 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
GUCY1A1 Q02108 1/20 0.35
GUCY1B1 Q02153 1/20 0.35
AR P10275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043739 0.79 ALDH1A1 (0.54) KMT2APCK1MEN1ALDH1A1DAO
SCHEMBL7417864 0.74 HCAR1 (0.42) KMT2AHCAR1MEN1ALDH1A1HPGD
SCHEMBL9235490 0.72 PNP (0.67) PNP
SCHEMBL7416425 0.71 PNP (0.47) KMT2AMEN1HPGDPNPMAPT
SCHEMBL7423403 0.69 KMT2A (0.48) KMT2AMEN1ALDH1A1PNPMAPT
SCHEMBL7604058 0.68 PNP (0.51) KMT2ADAOPNPMAPT
SCHEMBL28043744 0.68 CYP1A2 (0.52) KMT2AMEN1ALDH1A1HPGDMAPT
SCHEMBL8422905 0.67 KMT2A (0.42) KMT2AMEN1ALDH1A1HPGDMAPT
SCHEMBL7422829 0.67 PNP (0.49) KMT2AMEN1ALDH1A1HPGDPNP
SCHEMBL28043741 0.66 KMT2A (0.50) KMT2AMEN1ALDH1A1DAOMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825993-A1 XANTHINES AND THEIR THERAPEUTIC USE Chiroscience Limited (GB) 1998-03-04 EP claimed
WO-1996036638-A1 XANTHINES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO claimed